Hydroxy Varenicline

• Catalog No.: H995600
• CAS Number: 357424-21-6
• M. F.: C13H13N3O
• M. W.: 227.26182
• Storage: Refrigerator

SYNONYMS

• IUPAC name: 5,8,14-triazatetracyclo[10.3.1.0^2,^1^1.0^4,^9]hexadeca-2,4,6,8,10-pentaen-6-ol
• IUPAC Traditional name: 5,8,14-triazatetracyclo[10.3.1.0^2,^1^1.0^4,^9]hexadeca-2,4,6,8,10-pentaen-6-ol
• Synonyms: 1,6,7,8,9,10-Hexahydro-6,10-methano-2H-pyrazino[2,3-h][3]benzazepin-2-one

DATABASE IDS

• CAS Number: 357424-21-6

PROPERTIES

• Apperance: Pale Yellow Solid
• Melting Point: 292-294°C
• Solubility: DMSO
• Solubility: Aqueous Acid
• Storage Condition: Refrigerator

DETAILS

Description (English)

A metabolite of Varenicline. Metabolite M3b.

REFERENCES

• Dow, J., et al.: Drug Metab. Dispos., 22, 738 (1994)
• Toide, K., et al.: Biochem. Pharmacol., 67, 1269 (1994)
• Coe, J., et al.: J. Med. Chem., 48, 3474 (1994)
• Doll, R., et al.: Br. J. Cancer, 92, 426 (1994)