4'-Hydroxy Trazodone β-D-Glucuronide Sodium Salt

• Catalog No.: H970025
• M. F.: C25H29ClN5NaO8
• M. W.: 585.96923
• Storage: Hygroscopic, Refrigerator, Under Inert Atmosphere

SYNONYMS

• IUPAC name: sodium (2R,3R,4R,5S,6R)-6-{2-chloro-4-[4-(3-{3-oxo-2H,3H-[1,2,4]triazolo[4,3-a]pyridin-2-yl}propyl)piperazin-1-yl]phenoxy}-3,4,5-trihydroxyoxane-2-carboxylate
• IUPAC Traditional name: sodium (2R,3R,4R,5S,6R)-6-{2-chloro-4-[4-(3-{3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl}propyl)piperazin-1-yl]phenoxy}-3,4,5-trihydroxyoxane-2-carboxylate
• Synonyms: 4-Hydroxytrazodone Glucuronide Sodium; 2-[3-[4-(m-Chloro-p-hydroxyphenyl)-1-piperazinyl]propyl]-s-triazolo[4,3-a]pyridin-3(2H)-one Glucuronide Sodium; 2-Chloro-4-[4-[3-(3-oxo-1,2,4-triazolo[4,3-a]pyridin-2(3H)-yl)propyl]-1-piperazinyl]phenyl β-D-Glucopyranosiduronic Acid Sodium

PROPERTIES

• Apperance: Off-White Solid
• Melting Point: 163-168°C (dec.)
• Solubility: DMSO
• Storage Condition: Hygroscopic, Refrigerator, Under Inert Atmosphere

DETAILS

Description (English)

A major glucuronide metabolite of Trazodone-HCl (T718500).

REFERENCES

• Yamato, C., et al.: Xenobiotica, 4, 765 (1974)