3β-Hydroxy Tibolone-13C,d3

• Catalog No.: H964262
• M. F.: C21H30O2
• M. W.: 315.45435484
• Storage: -20°C Freezer, Under Inert Atmosphere

SYNONYMS

• IUPAC name: (1S,5S,9S,10R,11S,14R,15S)-14-ethynyl-9-(^1^3C,^2H₃)methyl-15-methyltetracyclo[8.7.0.0^2,^7.0^1^1,^1^5]heptadec-2(7)-ene-5,14-diol
• IUPAC Traditional name: (1S,5S,9S,10R,11S,14R,15S)-14-ethynyl-9-(^1^3C,^2H₃)methyl-15-methyltetracyclo[8.7.0.0^2,^7.0^1^1,^1^5]heptadec-2(7)-ene-5,14-diol
• Synonyms: (3β,7α,17α)-7-(Methyl-13C,d3)-19-norpregn-5(10)-en-20-yne-3,17-diol-d4; (3β,7α,17α)-3,17-Dihydroxy-7-(methyl-13C,d3)-19-norpregn-5(10)-en-20-yl-3-one; Org 30126-13C,d3

PROPERTIES

• Apperance: White Solid
• Melting Point: 79-84°C
• Solubility: Chloroform
• Solubility: Ethyl Acetate
• Storage Condition: -20°C Freezer, Under Inert Atmosphere

DETAILS

Description (English)

A labelled metabolite of Tibolone. A synthetic steroid with weak estrogenic, androgenic and progestogenic activity. A pharamceutical used in the treatment of menopausal syndrome.

REFERENCES

• Belman, S., et al.: Cancer Res., 32, 450 (1972)
• Shirahashi, H., et al.: Chem. Pharm. Bull., 41, 1664 (1972)
• Hoyte, R., et al.: Steroids, 58, 13 (1972)
• Sandker, G., et al.: Xenobiotica, 24, 143 (1972)
• Colombo, D., et al.: Eur. J. Med. Chem., 40, 69 (20