N-Desethyl Vardenafil-d8

• Catalog No.: D289952
• M. F.: C21H28N6O4S
• M. W.: 460.54982
• Storage: -20°C Freezer

SYNONYMS

• IUPAC name: 2-{2-ethoxy-5-[(2,2,3,3,5,5,6,6-^2H₈)piperazine-1-sulfonyl]phenyl}-5-methyl-7-propyl-3H,4H-imidazo[4,3-f][1,2,4]triazin-4-one
• IUPAC Traditional name: 2-{2-ethoxy-5-[(2,2,3,3,5,5,6,6-^2H₈)piperazine-1-sulfonyl]phenyl}-5-methyl-7-propyl-3H-imidazo[4,3-f][1,2,4]triazin-4-one
• Synonyms: 1-[[3-(1,4-Dihydro-5-methyl-4-oxo-7-propylimidazo[5,1-f][1,2,4]triazin-2-yl)-4-ethoxyphenyl]sulfonyl]-piperazine-d8

PROPERTIES

• Apperance: White Solid
• Melting Point: 94-97°C
• Solubility: DMSO
• Solubility: Methanol
• Storage Condition: -20°C Freezer

DETAILS

Description (English)

A Labelled metabolite of Vardenafil, a phosphodiesterase 5 inhibitor.

REFERENCES

• Bischoff, E., et al.: J. Urol., 165, 1316 (2001)
• Kim, N.N., et al.: Life Sci., 69, 2249 (2001)
• Kendirci, M., et al.: Expert Opin. Pharmacother., 5, 923 (2001)