8-CYCLOPENTYL-1,3-DIMETHYLXANTHINE

• Catalog No.: C988490
• CAS Number: 35873-49-5
• M. F.: C12H16N4O2
• M. W.: 248.28104
• Storage: -20°C Freezer

SYNONYMS

• IUPAC name: 8-cyclopentyl-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
• IUPAC Traditional name: 8-cyclopentyl-1,3-dimethyl-7H-purine-2,6-dione
• Synonyms: 8-Cyclopentyl-3,9-dihydro-1,3-dimethyl-1H-purine-2,6-dione; CPT, NSC 101806; 8-Cyclopentyltheophylline

DATABASE IDS

• CAS Number: 35873-49-5

PROPERTIES

• Apperance: White to Off-White Solid
• Melting Point: 250-252°C
• Solubility: DMSO
• Solubility: 0.1N Sodium Hydroxide
• Solubility: Water (<0.28 mg/ml)
• Storage Condition: -20°C Freezer

DETAILS

Description (English)

A selective A1 adenosine receptor antagonist. Binding activity in rat brain membranes: Ki = 10.9 nM (A1 receptor); Ki = 1440 nM (A2 receptor).

REFERENCES

• Klaasse, E., et al.: Eur. J. Pharmacol., 499, 91 (2004)
• Romanelli, L., et al.: Neurotoxicol., 26, 829 (2004)
• Rezvani, M.E., et al.: Can. J. Physiol. Pharmacol., 85, 606 (2004)