Centchroman-d6

• Catalog No.: C256602
• M. F.: C30H35NO3
• M. W.: 457.6038

SYNONYMS

• IUPAC name: 1-(2-{4-[(3S,4S)-7-methoxy-2,2-bis(^2H₃)methyl-3-phenyl-3,4-dihydro-2H-1-benzopyran-4-yl]phenoxy}ethyl)pyrrolidine
• IUPAC Traditional name: 1-(2-{4-[(3S,4S)-7-methoxy-2,2-bis(^2H₃)methyl-3-phenyl-3,4-dihydro-1-benzopyran-4-yl]phenoxy}ethyl)pyrrolidine
• Synonyms: trans-Centchroman; 3,4-trans-2,2-(Dimethyl-d6)-3-phenyl-4-[p-(β-pyrrolidinoethoxy)phenyl]-7-methoxychroman; rel-1-[2-[4-[(3R,4R)-3,4-Dihydro-7-methoxy-2,2-(dimethyl-d6)-3-phenyl-2H-1-benzopyran-4-yl]phenoxy]ethyl]pyrrolidine; Ormeloxifene; 1-[2-[p-(trans-7-Methoxy-2,2-(dimethyl-d6)-3-phenyl-4-chromanyl)phenoxy]ethyl]pyrrolidine; 67/20

DETAILS

Description (English)

Labelled Centchroman (C256600). Centchroman is an estrogen antagonist. Centchroman is a synthetic nonsteroidal postcoital antifertility agent.

REFERENCES

• Saeed, A., et al.: J. Med. Chem., 33, 3210 (1990)
• Richard, J., et al.: Drug Metab. Dispos., 28, 503 (1990)
• Delmas, P., et al.: Lancet, 359, 2018 (1990)
• Makker, A., et al.: Fertil Steril, 91, 2298 (1990)