(S)-Bicalutamide-d4

• Catalog No.: B382012
• M. F.: C24H22F4N2O10S
• M. W.: 606.4974928
• Storage: -20°C Freezer

SYNONYMS

• IUPAC name: (2S,3S,4S,5R,6S)-6-(1-{[4-cyano-3-(trifluoromethyl)phenyl]carbamoyl}-2-(4-fluorobenzenesulfonyl)-1-methylethoxy)-3,4,5-trihydroxyoxane-2-carboxylic acid
• IUPAC Traditional name: (2S,3S,4S,5R,6S)-6-(1-{[4-cyano-3-(trifluoromethyl)phenyl]carbamoyl}-2-(4-fluorobenzenesulfonyl)-1-methylethoxy)-3,4,5-trihydroxyoxane-2-carboxylic acid
• Synonyms: (2S)-N-[4-Cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluorophenyl-d4)sulfonyl]-2-hydroxy-2-methylpropanamide; (S)-Casodex-d4

PROPERTIES

• Apperance: Off-White Crystalline Solid
• Melting Point: 175-179°C
• Solubility: Acetone
• Solubility: Ethyl Acetate
• Storage Condition: -20°C Freezer

DETAILS

Description (English)

Labelled (S)-Enantiomer of Bicalutamide. Used as an antiandrogen, antineoplastic (hormonal).

REFERENCES

• Tucker, H., et al.: J. Med. Chem., 31, 954 (1988)
• Cockshott, I.D., et al.: Eur. Urol., 18, Suppl. 3, 10 (1988)
• Cockshott, I., et al.: Br. J. Clin. Pharm., 36, 339 (1988)
• McKillop, D., et al.: Xenobiotica, 25, 623 (1988)