Azasetron-13C,D3 Hydrochloride

• Catalog No.: A802803
• M. F.: C17H21Cl2N3O3
• M. W.: 387.26559484
• Storage: -20°C Freezer

SYNONYMS

• IUPAC name: N-{1-azabicyclo[2.2.2]octan-3-yl}-6-chloro-4-(^1^3C,^2H₃)methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-8-carboxamide hydrochloride
• IUPAC Traditional name: 6-chloro-4-(^1^3C,^2H₃)methyl-3-oxo-N-[(1s,4s)-1-azabicyclo[2.2.2]octan-3-yl]-2H-1,4-benzoxazine-8-carboxamide hydrochloride
• Synonyms: N-1-Azabicyclo[2.2.2]-oct-3-yl-6-chloro-3,4-dihydro-4-(methyl-13C,d3)-3-oxo-2H-1,4-benzoxazine-8-carboxamide Hydrochloride

PROPERTIES

• Apperance: White Solid
• Melting Point: 271-275°C (dec.)
• Solubility: DMSO
• Solubility: Water
• Storage Condition: -20°C Freezer

DETAILS

Description (English)

A 5-HT3 receptor antagonist. Used as an antiemetic.

REFERENCES

• Sato, N., et al.: Japan J. Pharmacol., 59, 443 (1992)
• Haga, K., et al.: Japan J. Pharmacol., 63, 377 (1993)