Azamulin

• Catalog No.: A801530
• CAS Number: 76530-44-4
• M. F.: C24H38N4O4S
• M. W.: 478.64792
• Storage: -20°C Freezer

SYNONYMS

• IUPAC name: 4-ethyl-3-hydroxy-2,4,7,14-tetramethyl-9-oxotricyclo[5.4.3.0^1,^8]tetradecan-6-yl 2-[(5-amino-4H-1,2,4-triazol-3-yl)sulfanyl]acetate
• IUPAC Traditional name: 4-ethyl-3-hydroxy-2,4,7,14-tetramethyl-9-oxotricyclo[5.4.3.0^1,^8]tetradecan-6-yl 2-[(5-amino-4H-1,2,4-triazol-3-yl)sulfanyl]acetate
• Synonyms: 14-O-(5-(2-Amino1,3,4-triazolyl)thioacetyl)dihydromutilin; SA 85530b; Antibiotic TDM 85-530

DATABASE IDS

• CAS Number: 76530-44-4

PROPERTIES

• Apperance: White to Off-White Solid
• Melting Point: >128°C (dec.)
• Solubility: DMSO
• Solubility: Methanol
• Storage Condition: -20°C Freezer

DETAILS

Description (English)

It is a highly selective human CYP3A4 inhibitor. A mutilin derivative.

REFERENCES

• Ballard, S., et al.: Biochem. Pharmacol., 37, 4643 (1988)
• Baldwin, S., et al.: Xenobiotica, 25, 261 (1988)
• Chiba, M., et al.: Biochem. Pharmacol., 62, 773 (1988)
• Bjornsson, T., et al.: Drug Metab. Dispos., 31, 815 (1988)