Asenapine-13C,d3

• Catalog No.: A788002
• M. F.: C17H16ClNO
• M. W.: 286.76069484
• Storage: -20°C Freezer, Under Inert Atmosphere

SYNONYMS

• IUPAC name: (2R,6R)-9-chloro-4-(^1^3C,^2H₃)methyl-13-oxa-4-azatetracyclo[12.4.0.0^2,^6.0^7,^1^2]octadeca-1(14),7(12),8,10,15,17-hexaene
• IUPAC Traditional name: (2R,6R)-9-chloro-4-(^1^3C,^2H₃)methyl-13-oxa-4-azatetracyclo[12.4.0.0^2,^6.0^7,^1^2]octadeca-1(14),7(12),8,10,15,17-hexaene
• Synonyms: trans-5-Chloro-2,3,3a,12b-tetrahydro-2-(methyl-13C,d3)-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole; (3aR,12bR)-rel-5-Chloro-2,3,3a,12b-tetrahydro-2-(methyl-13C,d3)-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole

PROPERTIES

• Apperance: Yellow Oil
• Solubility: Chloroform
• Solubility: Dichloromethane
• Storage Condition: -20°C Freezer, Under Inert Atmosphere

DETAILS

Description (English)

Combined serotonin (5HT2) and dopamine (D2) receptor antagonist; structurally related to labelled Mianserin. Antipsychotic.

REFERENCES

• Meltzer, H., et al.: J. Pharmacol. Exp. Ther., 251, 238 (1989)
• Schotte, A., et al.: Brain Res., 631, 191 (1989)
• Andree, B., et al.: Psychopharmacology, 131, 339 (1989)
• Richelson, E., et al.: Life Sci., 68, 29 (1989)