[D-Pen2,5]-Enkephalin hydrate

• Catalog No.: E3888
• M. F.: C30H39N5O7S2
• M. W.: 645.78996
• Purity: ≥95% (HPLC)

SYNONYMS

• IUPAC name: (4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-7-benzyl-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triazacyclotetradecane-4-carboxylic acid
• IUPAC Traditional name: (4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-7-benzyl-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triazacyclotetradecane-4-carboxylic acid
• Synonyms: DPDPE

DATABASE IDS

• MDL Number: MFCD00076430

PROPERTIES

• Empirical Formula (Hill Notation): C30H39N5O7S2 · xH2O
• Purity: ≥95% (HPLC)
• Personal Protective Equipment: Eyeshields, Gloves, type N95 (US), type P1 (EN143) respirator filter
• Storage Temperature: -20°C
• German water hazard class: 3

DETAILS

Description (English)

Amino Acid Sequence
Tyr-Pen-Gly-Phe-Pen [Disulfide Bridge: 2-5]
Biochem/physiol Actions
Antinociceptive activity mediated through the δ1 receptor while the modulatory activity is mediated through the δ2 receptor. Tritiated [D-Pen2,5]-enkephalin is used as a δ1 ligand.

Description (简体中文)

Amino Acid Sequence
Tyr-Pen-Gly-Phe-Pen [Disulfide Bridge: 2-5]
Biochem/physiol Actions
Antinociceptive activity mediated through the δ1 receptor while the modulatory activity is mediated through the δ2 receptor. Tritiated [D-Pen2,5]-enkephalin is used as a δ1 ligand.