CPA 1 hydrate

• Catalog No.: SML0125
• CAS Number: 111258-00-5(anhydrous)
• M. F.: C16H10O7
• M. W.: 314.2464
• Purity: ≥98% (HPLC)

SYNONYMS

• IUPAC name: 5,14-dioxatetracyclo[7.7.0.0^2,^6.0^1^1,^1^5]hexadeca-1,3,6,8,10,12,15-heptaene-4,13-dicarboxylic acid hydrate
• IUPAC Traditional name: 5,14-dioxatetracyclo[7.7.0.0^2,^6.0^1^1,^1^5]hexadeca-1,3,6,8,10,12,15-heptaene-4,13-dicarboxylic acid hydrate
• Synonyms: Naphtho[2,1-b:7,6-b′]difuran-2,8-dicarboxylic acid hydrate; NSC 623721 hydrate

DATABASE IDS

• MDL Number: MFCD20488061
• CAS Number: 111258-00-5(anhydrous)

PROPERTIES

• Empirical Formula (Hill Notation): C16H8O6 · xH2O
• Purity: ≥98% (HPLC)
• Apperance: gray-brown powder
• Solubility: DMSO: ≥15 mg/mL
• Storage Temperature: 2-8°C

DETAILS

Description (English)

Biochem/physiol Actions
CPA 1 is a potent, selective, ATP-competitive dual inhibitor of protein kinase casein kinase 2 (CK2) and proviral insertion Moloney virus kinases (Pim kinases). CPA 1 is selective for CK2 and Pim kinases (Pim-1, Pim-2, and Pim-3) when evaluated against a panel of 112 protein kinases.

Description (简体中文)

Biochem/physiol Actions
CPA 1 is a potent, selective, ATP-competitive dual inhibitor of protein kinase casein kinase 2 (CK2) and proviral insertion Moloney virus kinases (Pim kinases). CPA 1 is selective for CK2 and Pim kinases (Pim-1, Pim-2, and Pim-3) when evaluated against a panel of 112 protein kinases.