1-Azakenpaullone

• Catalog No.: A3734
• CAS Number: 676596-65-9
• M. F.: C15H10BrN3O
• M. W.: 328.1634
• Purity: ≥97% (HPLC)
• Storage: protect from light

SYNONYMS

• IUPAC name: 14-bromo-3,8,18-triazatetracyclo[9.7.0.0^2,^7.0^1^2,^1^7]octadeca-1(11),2(7),3,5,12,14,16-heptaen-9-one
• IUPAC Traditional name: 14-bromo-3,8,18-triazatetracyclo[9.7.0.0^2,^7.0^1^2,^1^7]octadeca-1(11),2(7),3,5,12,14,16-heptaen-9-one
• Synonyms: 9-Bromo-7,12-dihydro-pyrido[3′,2′:2,3]azepino[4,5-b]indol-6(5H)-one

DATABASE IDS

• MDL Number: MFCD09037522
• CAS Number: 676596-65-9

PROPERTIES

• Empirical Formula (Hill Notation): C15H10BrN3O
• Purity: ≥97% (HPLC)
• Apperance: gray-brown powder
• Solubility: DMSO: >10 mg/mL
• Storage Condition: protect from light
• Storage Temperature: 2-8°C
• German water hazard class: 2

DETAILS

Description (English)

Caution
air sensitive
Biochem/physiol Actions
1-Azakenpaullone is a cell permeable, potent, selective inhibitor of glycogen synthase kinase 3β (GSK3β) with 100-fold less cross-reactivity against CDKs. 1-Azakenpaullone can be used together with BIO and CHIR99021 as "gold standards" for GSK3 inhibition.

Description (简体中文)

Caution
air sensitive
Biochem/physiol Actions
1-Azakenpaullone is a cell permeable, potent, selective inhibitor of glycogen synthase kinase 3β (GSK3β) with 100-fold less cross-reactivity against CDKs. 1-Azakenpaullone can be used together with BIO and CHIR99021 as "gold standards" for GSK3 inhibition.