[des-Gly9-β-Mercapto-β,β-cyclopentamethylenepropionyl1,O-Et-Tyr2,Val4,Arg8]-Vasopressin

• Catalog No.: V4503
• CAS Number: 90332-81-3
• M. F.: C51H74N12O10S2
• M. W.: 1079.33766
• Purity: ≥97% (HPLC)

SYNONYMS

• IUPAC name: (2S)-2-{[(2S)-1-[(10R,13S,16S,19S,22S)-19-benzyl-13-(carbamoylmethyl)-22-[(4-ethoxyphenyl)methyl]-12,15,18,21,24-pentaoxo-16-(propan-2-yl)-7,8-dithia-11,14,17,20,23-pentaazaspiro[5.19]pentacosane-10-carbonyl]pyrrolidin-2-yl]formamido}-5-carbamimidamidopentanamide
• IUPAC Traditional name: (2S)-2-{[(2S)-1-[(10R,13S,16S,19S,22S)-19-benzyl-13-(carbamoylmethyl)-22-[(4-ethoxyphenyl)methyl]-16-isopropyl-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaazaspiro[5.19]pentacosane-10-carbonyl]pyrrolidin-2-yl]formamido}-5-carbamimidamidopentanamide
• Synonyms: (d(CH2)51, Tyr(Et)2, Val4, Arg8, des-Gly-NH29)-Vasopressin

DATABASE IDS

• MDL Number: MFCD00076750
• CAS Number: 90332-81-3

PROPERTIES

• Empirical Formula (Hill Notation): C51H74N12O10S2
• Purity: ≥97% (HPLC)
• GHS Signal Word: Warning
• GHS Hazard statements: H332
• European Hazard Symbols: Harmful (Xn)
• Personal Protective Equipment: dust mask type N95 (US), Eyeshields, Gloves
• Risk Statements: 20
• Safety Statements: 36
• Storage Temperature: -20°C
• German water hazard class: 3

DETAILS

Description (English)

Amino Acid Sequence
(1-Mercaptocyclohexyl)acetyl-Tyr(O-Ethyl)-Phe-Val-Asn-Cys-Pro-Arg-NH2 [Disulfide Bridge: 1-6]
Biochem/physiol Actions
Potent V1 (vasopressor) and V2 (antidiuretic) vasopressin receptor antagonist.

Description (简体中文)

Amino Acid Sequence
(1-Mercaptocyclohexyl)acetyl-Tyr(O-Ethyl)-Phe-Val-Asn-Cys-Pro-Arg-NH2 [Disulfide Bridge: 1-6]
Biochem/physiol Actions
Potent V1 (vasopressor) and V2 (antidiuretic) vasopressin receptor antagonist.