PG01037 dihydrochloride hydrate

• Catalog No.: SML0018
• CAS Number: 675599-62-9(anhydrous)
• M. F.: C26H30Cl4N4O2
• M. W.: 572.354
• Purity: ≥98% (HPLC)

SYNONYMS

• IUPAC name: N-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-en-1-yl}-4-(pyridin-2-yl)benzamide hydrate dihydrochloride
• IUPAC Traditional name: N-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-en-1-yl}-4-(pyridin-2-yl)benzamide hydrate dihydrochloride
• Synonyms: N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-(pyridin-2-yl)benzamide dihydrochloride hydrate; N-[(2E)-4-[4-(2,3-Dichlorophenyl)-1-piperazinyl]-2-buten-1-yl]-4-(2-pyridyl)benzamide dihydrochloride hydrate

DATABASE IDS

• MDL Number: MFCD20527309
• CAS Number: 675599-62-9(anhydrous)

PROPERTIES

• Empirical Formula (Hill Notation): C26H26Cl2N4O · 2HCl · xH2O
• Purity: ≥98% (HPLC)
• Apperance: white to tan powder
• Solubility: H2O: ≥8 mg/mL at ~60 °C
• Storage Temperature: 2-8°C

DETAILS

Description (简体中文)

Biochem/physiol Actions
PG01037 dihydrochloride is a selective dopamine D3 receptor antagonist. It is more selective for D3 receptors than other D3 antagonists that are currently available with a D2/D3 selectivity ratio of 867and a D4/D3 selectivity ratio of 13,000.
Selective dopamine D3 receptor antagonist