Pirenperone

• Catalog No.: P126
• CAS Number: 75444-65-4
• M. F.: C23H24FN3O2
• M. W.: 393.4539632
• Purity: >97%

SYNONYMS

• IUPAC name: 3-{2-[4-(4-fluorobenzoyl)piperidin-1-yl]ethyl}-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
• IUPAC Traditional name: pirenperone
• Synonyms: R-47,465; 3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2-methyl-4H-pyrido-[1,2-a] pyrimidin-4-one

DATABASE IDS

• PubChem SID: 24278110
• CAS Number: 75444-65-4
• EC Number: 278-213-5
• MDL Number: MFCD00069332

PROPERTIES

• Purity: >97%
• Gene Information: human ... HTR2A(3356), HTR2B(3357), HTR2C(3358)
• Apperance: light yellow solid
• Solubility: 0.1 M HCl: soluble11 mg/mL
• Solubility: methanol: soluble2.5 mg/mL
• Solubility: 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: soluble5.0 mg/mL
• Personal Protective Equipment: Eyeshields, Gloves, type N95 (US), type P1 (EN143) respirator filter
• German water hazard class: 3

DETAILS

Description (English)

Biochem/physiol Actions
5-HT2 serotonin receptor antagonist.
Other Notes
Tandem Mass Spectrometry data independently generated by Scripps Center for Metabolomics is available to view or download in PDF. P126.pdf Tested metabolites are featured on Scripps Center for Metabolomics METLIN Metabolite Database. To learn more, visit sigma.com/metlin.