Nα-Adamantaneacetyl-D-Arg-[Hyp3, Thi5,8, D-Phe7]-Bradykinin

• Catalog No.: B6029
• CAS Number: 130942-96-0
• M. F.: C68H99N19O14S2
• M. W.: 1470.76256
• Purity: ≥97% (HPLC)

SYNONYMS

• IUPAC name: (2S)-5-carbamimidamido-2-[(2S)-2-[(2R)-2-[(2S)-2-[(2S)-2-(2-{[(2S,4R)-1-[(2S)-1-[(2S)-5-carbamimidamido-2-[(2R)-5-carbamimidamido-2-{2-[(3R,5S,7s)-adamantan-1-yl]acetamido}pentanamido]pentanoyl]pyrrolidine-2-carbonyl]-4-hydroxypyrrolidin-2-yl]formamido}acetamido)-3-(thiophen-2-yl)propanamido]-3-hydroxypropanamido]-3-phenylpropanamido]-3-(thiophen-2-yl)propanamido]pentanoic acid
• IUPAC Traditional name: (2S)-5-carbamimidamido-2-[(2S)-2-[(2R)-2-[(2S)-2-[(2S)-2-(2-{[(2S,4R)-1-[(2S)-1-[(2S)-5-carbamimidamido-2-[(2R)-5-carbamimidamido-2-{2-[(3R,5S,7s)-adamantan-1-yl]acetamido}pentanamido]pentanoyl]pyrrolidine-2-carbonyl]-4-hydroxypyrrolidin-2-yl]formamido}acetamido)-3-(thiophen-2-yl)propanamido]-3-hydroxypropanamido]-3-phenylpropanamido]-3-(thiophen-2-yl)propanamido]pentanoic acid

DATABASE IDS

• CAS Number: 130942-96-0
• MDL Number: MFCD00142579

PROPERTIES

• Purity: ≥97% (HPLC)
• Gene Information: human ... BDKRB2(624)mouse ... BDKRB2(12062)rat ... BDKRB2(25245)
• Personal Protective Equipment: Eyeshields, Gloves, type N95 (US), type P1 (EN143) respirator filter
• Storage Temperature: -20°C
• German water hazard class: 3

DETAILS

Description (English)

Amino Acid Sequence
Nα-Adamantaneacetyl-D-Arg-Arg-Pro-Hydroxy-Pro-Gly-β-(2-Thienyl)Ala-Ser-D-Phe-β-(2-Thienyl)Ala-Arg
Biochem/physiol Actions
A highly potent antagonist at bradykinin B2 receptors with no agonist activity.