Oxycodone

• Catalog No.: Oxycodone
• CAS Number: 76-42-6
• M. F.: C18H21NO4
• M. W.: 315.36364

SYNONYMS

• IUPAC name: (1S,5R,13R,17S)-17-hydroxy-10-methoxy-4-methyl-12-oxa-4-azapentacyclo[9.6.1.0^1,^1^3.0^5,^1^7.0^7,^1^8]octadeca-7,9,11(18)-trien-14-one
• IUPAC Traditional name: oxycodone
• Brand Name: Oxycodone
• Synonyms: dihydrohydroxycodeinone; 14-hydroxydihydrocodeinone; 6-deoxy-7,8-dihydro-14-hydroxy-3-O-methyl-6-oxomorphine

DATABASE IDS

• CHEMBL: 656
• Wikipedia Title: Oxycodone
• CHEBI ID: 7852
• Chemspider ID: 4447649
• CAS Number: 76-42-6
• ATC CODE: N02AA05
• KEGG ID: D05312
• Medline Plus: a682132
• PubChem CID: 5284603
• ATC CODE: N02AA55
• DrugBank ID: DB00497
• Unique Ingredient Identifier: CD35PMG570

PROPERTIES

• Admin Routes: oral, intramuscular, intravenous, intranasal, subcutaneous, transdermal, rectal, epidural
• Bioavailability: 100% (IV); Up to 87% (oral)
• Dependency Liability: Moderate–High
• Excretion: Urine (19% unchanged)
• Half Life: 3–4.5 h
• Legal Status: Schedule 8 (Australia)
• Legal Status: Schedule I (Canada)
• Legal Status: Class A (CD)Schedule II (UK)
• Legal Status: Schedule II (US)
• Metabolism: Hepatic: primarily CYP3A, secondarily CYP2D6
• Pregnancy Category: B/D (prolonged use or in high doses at term)
• Protein Bound: 45%
• Solubility: HCl: 166 mg/mL (20°C)