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(4S)-1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-(3-chloro-4-fluorophenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
2-(3-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
1-{2-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)ethyl]piperidin-1-yl}propan-1-one
N-tert-butyl-3-[2-(3,4-dichlorophenyl)morpholin-4-yl]propanamide
1-(2-{2-azaspiro[4.4]nonan-2-ylmethyl}-4-methoxyphenoxy)-3-(dimethylamino)propan-2-ol
1-[(2-chloro-6-fluorophenyl)methyl]-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
1-(5-methyl-1H-pyrazole-3-carbonyl)-3-(naphthalene-1-carbonyl)piperidine
(2S,4S)-4-amino-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-N-methylpyrrolidine-2-carboxamide
(1R,5S)-6-[5-(3-methoxyphenyl)-1,2,4-triazin-3-yl]-6-azabicyclo[3.2.1]octane
N,N-dimethyl-5-{[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-1,3-thiazol-2-amine
(3aS,6aS)-2-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-{[(cyclopentylmethyl)(methyl)amino]methyl}-6-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
2-(5-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-methyl-1H-1,2,4-triazol-1-yl)ethan-1-ol
6-methyl-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-oxo-4H-pyran-2-carboxamide
1-(6-methylquinolin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(dimethyl-1,2-oxazol-4-yl)-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)acetamide
N-(1-{2-methyl-2,8-diazaspiro[4.5]decane-3-carbonyl}piperidin-4-yl)pyrimidin-2-amine
N-cyclopentyl-2-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
4-(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)-1,4-oxazepane
3-(3-methyl-1H-pyrazol-1-yl)-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]propanamide
1-[1-(3,4-dichlorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
3-[2-(dimethylamino)-N-methyl-2-(4-methylphenyl)acetamido]-N-methylpropanamide
methyl 3-(2-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)propanoate
1-ethyl-N-[2-(piperidin-1-yl)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(4-fluorophenyl)methyl]-3-(2-methoxybenzoyl)piperidine
2-(dimethyl-1,2-oxazol-4-yl)-N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)acetamide
1-(4,7-dimethylquinazolin-2-yl)-N-(thiophen-3-ylmethyl)piperidine-4-carboxamide
(2S,4R)-4-amino-1-[(3-ethoxy-2-hydroxyphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[3-(methylsulfanyl)propanoyl]piperidine-2-carboxamide
4-({4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)phenol
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(3-fluorophenyl)-1,3-benzoxazole-5-carboxamide
5-{1-[3-(thiophen-2-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-[(2-methylnaphthalen-1-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-ethyl-4-{2-[3-(2-methylphenyl)piperidin-1-yl]-2-oxoethyl}piperazine-2,3-dione
7-(2-hydroxyethyl)-2-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
(1R,3S,5S)-8-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
N-ethyl-3-[(4-fluorophenyl)formamido]-N-(pyridin-4-ylmethyl)propanamide
3-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-(methylsulfanyl)pyridine
[(2-chloro-4-fluorophenyl)methyl][(5-cyclopropyl-1,2-oxazol-3-yl)methyl]methylamine
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[1-(7-chloroquinoxalin-2-yl)piperidin-3-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-4-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-6-(propan-2-yl)pyrimidine
1-cyclopentyl-4-(6-ethyl-2-methylquinoline-4-carbonyl)piperazin-2-one
2-{1-[(4-fluorophenyl)methyl]-4-(6-phenylpyridazin-3-yl)piperazin-2-yl}ethan-1-ol
S-(2-acetyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-N-benzyl-1-hydroxypropane-2-sulfonamido
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-{imidazo[1,2-a]pyridin-3-yl}ethan-1-one
6-tert-butyl-2-(3-{[methyl(pyrimidin-4-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperazine
1-(3-chloro-5-methoxybenzoyl)-N,N-dimethylazepan-4-amine