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N-[3-(4-{[3-(2H-1,3-benzodioxol-5-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide
1-(3-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-3-oxopropyl)piperidin-2-one
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-(3-hydroxypropyl)-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
2-{4-[(2,3-difluorophenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
1-{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}piperidine-4-carboxamide
7-{[2-(benzylamino)pyrimidin-5-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(4-{[(3-phenoxyphenyl)carbamoyl]amino}piperidin-1-yl)acetamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]ethan-1-one
1-cycloheptyl-4-[(1-methylpiperidin-4-yl)amino]pyrrolidin-2-one
2-({4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)benzoic acid
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethylfuran-3-carboxamide
N,N-dimethyl-3-[3-(2-methylphenyl)piperidine-1-carbonyl]aniline
(3S,4S)-N-(3-cyano-4-methoxyphenyl)-3-hydroxy-4-(morpholin-4-yl)pyrrolidine-1-carboxamide
2-(4-{[3-(2-hydroxyethoxy)phenyl]methyl}morpholin-3-yl)acetic acid
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-{5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(morpholin-4-yl)propan-1-one
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
1,3,6-trimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-4-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
1-{6-methyl-5-[5-(1-methylpiperidin-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}butan-1-one
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
6-(2-fluoro-4-methoxyphenyl)-N-[(2S)-2-hydroxypropyl]-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
3,3-dimethyl-1-{[5-(3-phenylbutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
3-{[(5-methylthiophen-2-yl)methyl]({[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl})amino}propan-1-ol
N-{[4-fluoro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(furan-2-yl)benzamide
8-[(2-aminopyridin-3-yl)methyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[2-(2-fluorophenyl)acetyl]-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[7-fluoro-2-(1H-pyrazol-4-yl)quinoline-4-carbonyl]piperidine-3-carbonitrile
2-{1-[(4-fluorophenyl)methyl]-4-(pyridin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-(1,2-benzoxazol-6-yl)-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methylurea
N-benzyl-3-[1-(2-chlorobenzenesulfonyl)piperidin-4-yl]-N-methylpropanamide
7-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(2-methoxyethyl)-1-methyl-5-[3-(pyridin-4-yl)azetidine-1-carbonyl]-1H-1,3-benzodiazol-2-amine
2-(3,4-dichlorophenyl)-4-(2,4-dimethylbenzoyl)morpholine
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]propan-1-one
1-methyl-2-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,2-dihydroquinoline-4-carboxamide
2-(butan-2-ylsulfanyl)-5-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}pyrimidine
2-(2-hydroxyethyl)-9-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
N,N-dimethyl-2-{[2-(2-oxopyrrolidin-1-yl)propanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-ethyl-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl){[4-(propan-2-yl)phenyl]methyl}amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-methanesulfonylbenzamide
3-hydroxy-3-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(3-phenylpropyl)piperidin-2-one
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})methylamine
N-(2-{[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)acetamide