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1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]pentan-1-one
cyclohexyl[4-(furan-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
N-{[3-methyl-7-(1,2,5-thiadiazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
3-[4-({4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidin-1-yl]pyrazine-2-carbonitrile
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
5-methyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1,2-oxazole-4-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]propanamide
4-hydroxy-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(1R,3S)-7-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-7-azaspiro[3.5]nonane-1,3-diol
4-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-1-(4-fluorophenyl)butan-1-one
2-methyl-4-(4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperazin-1-yl)-5-propylpyrimidine
N-(1-phenylethyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
methyl[(4-methyl-1,3-thiazol-2-yl)methyl]{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
2-[(2-{1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
2-({4-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
5-[2-({8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}amino)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-(2-methylphenyl)-4-[(1-methylpyrrolidin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})(pyridin-2-ylmethyl)amine
5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}quinoxaline
2-chloro-4-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}phenol
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]pyridine-2-carboxamide
6-(benzyloxy)-1-cyclohexyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1,4-diazepan-2-one
4-(4-ethyl-2-methyl-1,3-thiazole-5-amido)-N-phenylpiperidine-1-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N,3-bis(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-(3-methylpiperidin-1-yl)-3-{[(4-phenyloxan-4-yl)methyl]amino}propan-1-one
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-[4-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepan-6-yl]oxy}acetamide
3-{1-[2-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}phenol
2-(4-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}piperazin-1-yl)-N-ethylacetamide
5,6-dimethyl-3-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
(3aS,6aR)-5-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
1-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-3-ol
4-methoxy-N-(2-methoxyethyl)-2-({1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)benzamide
2-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)-1,3-benzoxazole
1-(2-methoxyethyl)-8-{[5-(methoxymethyl)furan-2-yl]methyl}-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4S)-1-({[2-(2-methoxyphenyl)ethyl]carbamoyl}methyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
1-(2-methoxyphenyl)-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazin-2-one
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
7-cyclopropanecarbonyl-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{[5-(4-hydroxyphenyl)-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-3-(1,2-oxazolidin-2-yl)propanamide
methyl 5-[(1-methoxy-1-oxopropan-2-yl)amino]-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1,2-dimethyl-1H-indol-5-ol
2-(4-{[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
2-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]benzonitrile
3-({2-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-chloro-N-{2-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
N3-cyclohexyl-1-cyclopropyl-N5-[1-(6-methoxynaphthalen-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[(4aR,8aR)-7-(3-acetylbenzoyl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one