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4-methyl-5-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
4-benzyl-1-(1-methylazepane-2-carbonyl)piperidin-4-ol
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-3-phenylpropanamide
6-(methylsulfanyl)-N-(2,4,6-trimethylpyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
2-ethoxy-5-[2-(3-methylbutyl)pyrimidin-4-yl]benzoic acid
4-[4-(benzenesulfonyl)piperazine-1-carbonyl]-1-methylimidazolidin-2-one
3-{5-[2-(cyclopent-2-en-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-phenyl-7-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-cyclopropyl-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-2-(1H-pyrazol-1-yl)acetamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-4-(2-oxopyrrolidin-1-yl)benzamide
2-(3-chloro-4-hydroxyphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
1-(1-{[3-(2-aminoethyl)phenyl]methyl}piperidin-3-yl)-2-phenylethan-1-one
1-{2-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one
2-benzyl-8-(oxolane-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-(propan-2-yl)-1-{1-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-yl}piperidine-4-carboxamide
2-(4-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
methyl 3-(2-chlorobenzenesulfonamido)-5-{[2-(1,3-thiazol-4-yl)acetamido]methyl}benzoate
N-[(2S,4R,6R)-2-(2-chloro-6-methylphenyl)-6-(propan-2-yl)oxan-4-yl]acetamide
4-(furan-3-yl)-6-(morpholin-4-yl)pyrimidin-2-amine
[(4-methanesulfonylphenyl)methyl][(2-methylphenyl)methyl](prop-2-en-1-yl)amine
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(pyrimidin-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-methoxy-2-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-5-methoxyphenol
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-[2-(3-methoxyphenyl)pyrrolidin-1-yl]pyridine
(3R,5S)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amino]methyl}phenol
5-(5-methanesulfonyl-2-methylpyrimidin-4-yl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
ethyl 3-({3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}amino)propanoate
5-acetyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]thiophene-2-carboxamide
2-{[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]methyl}phenol
4-(methylsulfanyl)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
N,2-dimethyl-6-(piperidin-4-yl)-N-(thiophen-3-ylmethyl)pyrimidin-4-amine
5-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}quinoxaline
N-{[2-(2-phenylethynyl)phenyl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(2-amino-4-methylpyrimidine-5-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
3-[(4-{[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl](methyl)amino}-6-methylpyrimidin-2-yl)amino]phenol
3-[(2,4-dimethoxy-3-methylphenyl)methyl]-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl})methylamine
4-{2-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]ethyl}phenol
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(dimethyl-1,2-oxazol-4-yl)acetamide
1-(5-chloro-2-methylphenyl)-4-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
2-{1-cyclohexyl-5-[(dimethylamino)(3-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
2-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)-2,7-diazaspiro[4.5]decan-6-one
(2R)-2-cyclohexyl-1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-hydroxyethan-1-one
[2-(3,4-dichlorophenyl)pyridin-4-yl]methanol
(1S,5R)-3-(5-propylthiophene-3-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
8-[(3-methoxyphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid