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1-({1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
9-(6-aminopyridine-3-carbonyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
3-(1-{1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
2-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
2-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
5-(2-{4-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-oxoethyl)pyrrolidin-2-one
1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]azepane
(2S,4R)-4-(3-cyanobenzamido)-N-[(2-methyl-1H-indol-5-yl)methyl]pyrrolidine-2-carboxamide
N-ethyl-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
3-(4-chlorobenzoyl)-1-(dimethyl-1,2-oxazole-4-carbonyl)piperidine
2-(2-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
2-({[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]amino}methyl)-6-methylquinolin-4-ol
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(methylsulfanyl)acetamide
4-(8-methoxy-2-methylquinolin-5-yl)-6-(pyrrolidin-1-yl)pyrimidin-2-amine
2-{9-[(2,5-dimethylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
4-fluoro-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N,3-dimethylbenzamide
4-(5-methyl-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)piperazine-1-carbaldehyde
3-(azetidine-1-carbonyl)-N-[(3-methoxyphenyl)methyl]-N-methylbenzene-1-sulfonamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
3-[3-(1H-pyrazol-1-yl)phenyl]-5-(pyrrolidine-1-sulfonyl)benzoic acid
1-methyl-4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
N-{1-[1-(quinolin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
8-(4,6-dimethylpyrimidin-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-3-methylbutan-1-one
(4aS,8aR)-6-[5-(methoxymethyl)furan-2-carbonyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-5-chlorophenol
4-methyl-6-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]pyrimidin-2-amine
(3R,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazole
3-{2-[3-(2-{[(3,4-difluorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]-2-oxoethyl}-1,2,3-oxadiazol-3-ium-5-olate
2-{1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
(2S)-3-phenyl-2-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)propanamide
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
1-cyclopentyl-N-methyl-6-oxo-N-(quinoxalin-2-ylmethyl)piperidine-3-carboxamide
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[2-(methylsulfanyl)ethyl]propanamide
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
9-(morpholine-2-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-ethyl-6-methyl-N4-[1-(5-methylpyridin-2-yl)ethyl]pyrimidine-2,4-diamine
[3-(1H-1,2,3-benzotriazol-1-yl)propyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
1-ethyl-4-[1-(4-fluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
1-(2,3-dihydro-1-benzofuran-2-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
2,4-dimethoxy-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzamide
2-benzyl-8-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[3-(3-methylphenyl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
8-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1-oxa-8-azaspiro[4.5]decane
(4aS,7aR)-N-(3-cyanophenyl)-4-(2-methylpropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-chloro-N-(2-{3-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]phenoxy}propyl)benzamide
ethyl 4-[6-(5-methyl-1H-indole-2-carbonyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
1-[9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one