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N-ethyl-4-methyl-2-(4-methylpiperazin-1-yl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-ethyl-1H-imidazol-1-yl)acetamide
4-methoxy-N-methyl-3-{1H-pyrazolo[3,4-b]pyridin-1-yl}benzamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,5-dimethylbenzamide
2-cyclohexyl-5-{[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]methyl}pyrimidine
1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
N-ethyl-4-{[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]amino}piperidine-1-carboxamide
(4aR,7aS)-1-benzyl-4-(2-hydroxypyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({1-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-3-yl}methyl)acetamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methoxyethyl)-N-methylpyridin-2-amine
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-methyl-2-oxopentanamide
methyl 3-[(adamantan-1-ylformamido)methyl]-5-propanamidobenzoate
(4aS,7aR)-1-[2-(3,4-dichlorophenyl)acetyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(pyridin-3-yloxy)piperidin-1-yl]ethan-1-one
(3S,4S)-4-cyclopropyl-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidine-3-carboxylic acid
{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
(5-{[2-(3-fluorophenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}furan-2-yl)methanol
2-{[5-(3-cyclopropyl-1H-pyrazol-5-yl)-4-(2,4-difluorophenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
5,7-dimethyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
(4-benzylpiperidin-4-yl)methanol
4-[(2S)-2-amino-3-phenylpropanoyl]-1-(2-methoxyphenyl)piperazin-2-one
1-{2-[2-(3-chlorophenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(furan-2-ylmethyl)-N-methylpiperidine-4-carboxamide
ethyl 5-(isoquinoline-3-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(2R,6R)-4-(1,3-dihydroxypropan-2-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
methyl 1-{3-[(4-chlorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
N-(1,4-dioxan-2-ylmethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-(furan-2-yl)-2-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]ethane-1,2-dione
[(3-fluoro-2-methoxyphenyl)methyl](methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
2-(2-methoxyethyl)-N-(oxolan-3-yl)-1,3-benzoxazole-6-carboxamide
ethyl 1-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]piperidine-2-carboxylate
2-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
1-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]-4-(pyridin-4-yl)piperazine
N,2-diethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}pyrimidine-5-carboxamide
9-(5-ethyl-1H-pyrrole-2-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(2-chlorophenyl)methyl]-3-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
4-(4-aminopyridine-2-carbonyl)-1-(3-methoxyphenyl)-3-methylpiperazin-2-one
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
6-(2-methoxyphenyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
5-{3-[3-(2-methylphenoxymethyl)piperidin-1-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
(1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-[(4-fluorophenyl)methyl]piperidin-3-yl)methanol
N-cyclopropyl-3-(pyridin-4-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
8-fluoro-2-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]quinoline
3-(2,3-dihydro-1H-inden-2-yl)-5-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
5-{2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1,5-dimethyl-4-({4-[2-(oxolan-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one