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3-[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)amino]-N-(pyridin-3-yl)propanamide
{3-[(2-fluorophenyl)methyl]-1-(quinolin-2-ylmethyl)piperidin-3-yl}methanol
3-[(1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]pyridine
4-fluoro-N-[3-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)phenyl]benzene-1-sulfonamide
8-[(4-fluorophenyl)methyl]-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N'-(3-hydroxyphenyl)-N-{1-oxaspiro[4.4]nonan-3-yl}butanediamide
2-(4-acetylphenoxy)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]ethan-1-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-methyl-N-(oxolan-2-ylmethyl)furan-3-carboxamide
2-(2,5-dimethoxyphenyl)-5-methyl-4-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1,3-oxazole
methyl 5-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-3-(furan-2-amido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-butyl-1-methyl-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazin-2-one
9-(2-amino-6-methylpyrimidin-4-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-chlorophenyl)-6-[5-(methoxymethyl)furan-2-carbonyl]-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-cyclopentyl-N'-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}butanediamide
(3S,4S)-1-[(5-ethylpyridin-2-yl)methyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-ethyl-4-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-(2-hydroxyethyl)-N-(propan-2-yl)-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-[5-(propan-2-yl)-1,2-oxazol-3-yl]-N-[4-(1H-pyrazol-1-yl)phenyl]pyrrolidine-1-carboxamide
9-[2-(2,5-dimethylphenyl)acetyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(propan-2-yl)phenyl]-4-[3-(pyridin-2-yl)azetidine-1-carbonyl]pyrrolidin-2-one
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidine
methyl 3-[6-(cyclopropylmethoxy)-4-[(3-methoxyphenyl)methyl]-3-oxo-1,4-diazepane-1-carbonyl]benzoate
4'-butyl-1-(3-methylpentanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-methyl-3-(2-methylpropyl)-8-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(1-benzofuran-5-carbonyl)-2-ethyl-1-(propan-2-yl)piperazine
6-[(2-hydroxy-4-methoxyphenyl)methyl]-N-{[3-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
(1S,5R)-3-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methoxyethyl)-2-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[2-({5-[1-(piperidin-1-yl)ethyl]furan-2-yl}formamido)ethyl]acetamide
methyl 1-{[4-(naphthalene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-4-carboxylate
methyl 7-oxo-3-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1H-indole
1-(1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carbonyl)piperidine-3-carboxamide
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(cyclopropylmethyl)-4-(2,3-difluoro-4-methylbenzoyl)-2-(propan-2-yl)-1,4-diazepane
5-ethanesulfonamido-1-methyl-2-phenyl-N-[1-(thiophen-3-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
N,N-dimethyl-2-[(piperidin-3-yl)amino]ethane-1-sulfonamide
(4aR,7aS)-1-benzyl-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N1-ethyl-N2-[2-(4-methoxyphenyl)phenyl]pyrrolidine-1,2-dicarboxamide
2-{4-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
5-acetamido-1-ethyl-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-fluorophenyl)-1H-1,3-benzodiazole-7-carboxamide
3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]piperidin-2-one
(3R,4R)-1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-4-cyclopropyl-3-methylpiperidin-4-ol
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[3-(1H-pyrazol-1-yl)propyl]pyrimidine-5-carboxamide
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-4-(pyridin-4-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
3-[5-({[2-(dimethylamino)ethyl][(5-methylthiophen-2-yl)methyl]amino}methyl)thiophen-3-yl]prop-2-yn-1-ol