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3-{cyclopropyl[(4-hydroxy-3-methoxyphenyl)methyl]carbamoyl}benzoic acid
(4aR,8aR)-1-cyclopropanecarbonyl-6-(3-methylbutyl)-decahydro-1,6-naphthyridine
1-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-3-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
1-[1-(6-cyanopyridin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-ethoxy-5-[2-(3-methoxyphenoxymethyl)pyrimidin-4-yl]benzoic acid
N-(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylfuran-2-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
1-[3-oxo-3-(4-phenylazepan-1-yl)propyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(methoxymethyl)-5-({4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}methyl)pyrimidine
3-[(oxolan-3-ylmethyl)sulfamoyl]-N-(2-phenoxyethyl)benzamide
N-[4-(3-hydroxy-4-methoxybenzamido)phenyl]-5-methylfuran-2-carboxamide
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(4-propylpyrimidine-5-carbonyl)azocane
2-(2-chloro-4-{[2-(propan-2-yl)-2,5-dihydro-1H-pyrrol-1-yl]methyl}phenoxy)acetamide
2-{[(1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
1-ethyl-N-[3-(methylsulfanyl)propyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-(1-{2-[cyclopentyl(methyl)amino]acetyl}piperidin-3-yl)benzoic acid
ethyl 4-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-{4-[2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(3,4,5-trimethoxyphenyl)ethan-1-one
6-chloro-2-methyl-4-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoline
3-chloro-N-(2-methoxyethyl)-4-[(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)oxy]benzamide
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
5-[(4-ethylpiperazin-1-yl)methyl]-N-[2-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(2-methoxybenzoyl)-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazine
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-(pyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-cyclohexyl-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1H-pyrazole-4-carboxamide
6-cyclopentyl-2-methoxy-3-({[4-(methylsulfanyl)butan-2-yl]amino}methyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-3,3-diphenylpiperidine
N-[(2-methoxyphenyl)methyl]-2-(morpholin-2-yl)-N-propylacetamide
(4-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane-8-carbonyl}phenyl)methanol
3-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}-4H-chromen-4-one
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-methanesulfonyl-4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)piperidine
2-(dimethylamino)-N-{[4-(dimethylamino)oxan-4-yl]methyl}-2-(3-methylphenyl)acetamide
6-(4-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperazin-1-yl)-9H-purine
N-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]-2-(pyrrolidin-3-yl)benzamide
4-{1-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl}morpholine
2-(3-chloro-5-fluoro-4-methoxyphenyl)-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
(2R,6R)-4-[(3,5-difluoro-4-methoxyphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2S)-4-methyl-1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)propyl]-2-phenylpiperazine
4-(2-{1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]piperidin-2-yl}ethyl)phenol
3-(dimethyl-1,2-oxazol-4-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}propanamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-4,6-dimethylpyrimidin-2-amine
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})(propan-2-yl)amine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-1,2,3-benzotriazole-5-carboxamide
4-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-6-methoxy-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
[(3,5-dichloropyridin-4-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine