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N-(cyclohexylmethyl)-1-cyclopropyl-5-[3-(diethylamino)pyrrolidine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
(3S,4S)-1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-8-methoxy-4-methylquinoline
1-[(4-fluoro-2-methylphenyl)methyl]-N,N-dimethylazepan-4-amine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyrrolidine-1-sulfonamide
2-(3,4-dichlorophenyl)-4-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]morpholine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-1,3-thiazole-4-carboxamide
ethyl 4-{1-ethyl-3-[(3-methoxyphenyl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}piperidine-1-carboxylate
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(3-methylphenyl)methyl]benzamide
3-chloro-4-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}phenol
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidine
5-ethoxy-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)furan-2-carboxamide
5-methyl-N-{4-[2-(prop-2-en-1-ylsulfanyl)propanamido]phenyl}furan-3-carboxamide
8-[(3-hydroxy-6-methylpyridin-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]amino}-N-(propan-2-yl)acetamide
6-[1-(2-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-3-yl}methyl)acetamide
2-methyl-N-[2-(7-methyl-1H-indol-3-yl)ethyl]-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
4-phenyl-1-[1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]butan-1-one
1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
1-(4-{[4-(2-aminoethyl)phenyl]methyl}-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
9-[(2,3,4-trimethoxyphenyl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
(3S,4R)-1-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-(4-fluoro-2-methylphenyl)acetamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}ethan-1-one
4-[4-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamide
N-(2-{7-[4-(4-methoxyphenyl)butan-2-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(furan-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-(6,8-dimethylquinolin-4-yl)-4-hydroxypiperidine-4-carboxylic acid
1-{2-hydroxy-3-[3-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
4-{4-[(4,4-difluoropiperidin-1-yl)methyl]phenyl}-2-methylbutan-2-ol
1-[2-(azepan-1-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-2-(furan-2-yl)ethane-1,2-dione
(2S)-N2-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}pyrrolidine-1,2-dicarboxamide
(1R,5S,6R)-N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
2-{2-[1-(2-methylfuran-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
2-[2-(pyridin-2-yl)ethyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-1-carboxamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]acetic acid
1-(dimethyl-1,3-thiazole-5-carbonyl)-3-(2-fluorophenoxymethyl)piperidine
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-methoxypyridine-3-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(2-methoxybenzoyl)piperazin-1-yl]propan-1-one
3-methoxy-N-(3-methyl-1-{7-[2-(pyridin-2-ylsulfanyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)propanamide
4-fluoro-N-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzamide
methyl 3-[({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)sulfamoyl]thiophene-2-carboxylate
1-(1-cyclohexanecarbonylpiperidin-3-yl)-4-(2-methoxyphenyl)piperazine
1-{2-[1-benzyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(5S,9aS,9bS)-5-[(E)-2-(furan-2-yl)ethenyl]-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(1-benzothiophen-2-ylmethyl)({[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine