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1-(4-bromo-1,3-thiazol-2-yl)piperidin-4-ol
1-(4-bromo-1,3-thiazol-2-yl)piperazine
1-(4-bromo-1,3-thiazol-2-yl)piperidine
2-bromo-6-cyclohexylpyridine
1-(6-bromopyridin-2-yl)piperidin-4-ol
2-chloro-5-fluoropyrazine
2-(tert-butoxy)-5-chloropyrazine
2-bromo-6-(pyrrolidin-1-yl)pyrazine
4-chloropyrimidine-2-carbonitrile
4-chloro-6-methylpyrimidine-2-carbonitrile
4-chloro-2-(pyrrolidin-1-yl)pyrimidine
4,6-dichloro-2-(pyrrolidin-1-yl)pyrimidine
4,6-dichloro-2-(1H-pyrazol-1-yl)pyrimidine
4,6-dichloro-2-(piperazin-1-yl)pyrimidine
6-chloropyrimidine-4-carbonitrile
2-(tetramethyl-1,3,2-dioxaborolan-2-yl)-4-(trifluoromethyl)pyridine
4-chloro-2-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine
2-tert-butyl-6-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine
(6-tert-butylpyridin-2-yl)boronic acid
(6-cyclohexylpyridin-2-yl)boronic acid
[6-(morpholin-4-yl)pyridin-2-yl]boronic acid
[6-(piperidin-1-yl)pyridin-2-yl]boronic acid
[6-(pyrrolidin-1-yl)pyridin-2-yl]boronic acid
[6-(tert-butoxy)pyridin-2-yl]boronic acid
(2-methoxypyrimidin-4-yl)boronic acid
[2-(morpholin-4-yl)pyrimidin-4-yl]boronic acid
(2-cyano-6-methylpyrimidin-4-yl)boronic acid
(2-cyanopyrimidin-4-yl)boronic acid
(6-chloro-2-methoxypyrimidin-4-yl)boronic acid
[6-chloro-2-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]boronic acid
[6-chloro-2-(piperidin-1-yl)pyrimidin-4-yl]boronic acid
[6-(pyrrolidin-1-yl)pyrazin-2-yl]boronic acid
[6-(morpholin-4-yl)pyrazin-2-yl]boronic acid
[6-(piperidin-1-yl)pyrazin-2-yl]boronic acid
[6-chloro-2-(pyrrolidin-1-yl)pyrimidin-4-yl]boronic acid
(5-ethoxypyrazin-2-yl)boronic acid
(5-methoxypyrazin-2-yl)boronic acid
[5-(1H-pyrazol-1-yl)pyrazin-2-yl]boronic acid
[5-(pyrrolidin-1-yl)pyrazin-2-yl]boronic acid
[5-(piperidin-1-yl)pyrazin-2-yl]boronic acid
[5-(morpholin-4-yl)pyrazin-2-yl]boronic acid
2-(4-methylpiperidin-1-yl)-6-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine
2-ethoxy-6-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine
2-(propan-2-yloxy)-6-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine
N-cyclopropyl-6-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-amine
N-cyclobutyl-6-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-amine
N-cyclopentyl-6-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-amine
N-cyclohexyl-6-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-amine
4-methyl-1-[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1,3-thiazol-2-yl]piperidine
N-cyclopropyl-4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1,3-thiazol-2-amine