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3-(4-chlorophenyl)-5-(4-fluorobenzoyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
8-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(ethyl)(2-methylprop-2-en-1-yl)amine
1-methyl-4-[(5-phenylthiophen-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
6-(difluoromethyl)-2-(2-{[3-(hydroxymethyl)-3-methylpiperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]amine
5-(propan-2-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2,4-oxadiazol-3-amine
2-({4-[2-(1-hydroxyethyl)-1H-1,3-benzodiazol-5-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
(2R)-3-(benzyloxy)-2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propan-1-ol
N-ethyl-5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}pyrimidin-2-amine
2-[benzyl(ethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-methyl-3-(2-methylpropyl)-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-pyrazole
4-chloro-2-({[(3R,5S)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]amino}methyl)phenol
4-chloro-N-[(4-hydroxyphenyl)methyl]-1,5-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
6-methyl-5-[3-(1H-pyrazol-5-yl)phenyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(4-ethyl-1H-pyrazol-5-yl)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidine
6-chloro-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
1-(2-phenylethyl)-8-(pyridin-2-ylmethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(cyclobutylmethyl)-2-[2-(3-fluorophenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-{[2-(cyclopropylmethyl)-7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
(2S,4R)-4-amino-N-methyl-1-({[(2-methylphenyl)methyl]carbamoyl}methyl)pyrrolidine-2-carboxamide
1-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-3-ethylpiperazine
2,5-dimethyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pyrimidin-4-amine
7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-4-[(2-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
(3S,5R)-N3-butyl-N5-(4-fluorophenyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-chloro-1,3-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
6-[(4-methylazepan-1-yl)methyl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(methoxymethyl)-1-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperidine
2-amino-N-[2-(pyridin-2-yl)ethyl]-1,3-benzothiazole-5-carboxamide
N-[2-(4-methoxyphenyl)phenyl]-1-(oxan-4-yl)piperidine-3-carboxamide
3-(1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-2-yl)pyridine
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-(3-{thieno[2,3-d]pyrimidin-4-yl}phenyl)-1H-pyrazole
6-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-2-carbonitrile
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-6-methoxypyrimidin-4-amine
1-(carbamoylmethyl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-3-carboxamide
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-4-(piperidin-1-yl)butan-1-one
2-(5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-sulfonyl}thiophen-2-yl)pyridine
[(2-ethylpyrimidin-4-yl)methyl](methyl)[2-(oxan-4-yl)ethyl]amine
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
(3S,4S)-4-cyclopropyl-1-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)pyrrolidine-3-carboxylic acid
6-(2-chlorophenyl)-N-(oxan-3-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(3S,4R)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
7-[(2S)-2-amino-6-hydroxyhexanoyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(morpholin-4-yl)acetyl]pyrrolidine-3-carboxylic acid