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1-(2,3-dihydro-1H-inden-2-yl)-5-(furan-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
2-benzyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1,3-benzoxazole-5-carboxamide
2-(azocan-1-yl)-1-[3-(3-methoxyphenoxy)azetidin-1-yl]ethan-1-one
1-(1-benzothiophene-2-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(1R,2S)-N1-tert-butyl-N2-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}cyclohexane-1,2-dicarboxamide
5-{furo[3,2-c]pyridin-4-yl}-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[(4-fluorophenyl)methyl]-5-[4-(propan-2-yloxy)benzoyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
2-(4-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetamide
2-(2,4-dimethoxyphenyl)-3-(pyrrolidine-1-carbonyl)pyridine
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
3-{1-[2-(1H-1,3-benzodiazol-2-yl)acetyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
10-methoxy-5-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl){[6-(trifluoromethyl)pyridin-3-yl]methyl}amine
N-({1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}methyl)acetamide
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
methyl 3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
1-[(2-chloro-4-fluorophenyl)methyl]-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
ethyl 1-(1H-imidazol-2-ylmethyl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
3-({[3-(2,4-dimethylphenoxy)-2-hydroxypropyl]carbamoyl}amino)-2-methylbenzamide
1-{[3-(cyclopropylmethyl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
4-(2-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}ethyl)benzene-1-sulfonamide
2-[3-(2-fluorophenyl)-4-methyl-1H-pyrazol-1-yl]-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
4-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2,6-dimethylphenol
3-({[(1-ethyl-1H-imidazol-2-yl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-4-acetamido-N-(2-methoxyethyl)benzamide
1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(1H-pyrazol-1-yl)propan-1-one
1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
4-benzyl-3-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
(2E)-N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
4,4,4-trifluoro-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]butan-1-one
4-(4-methyl-1H-pyrazol-1-yl)-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidine-4-carboxylic acid
2-[1'-(5-methoxyfuran-2-carbonyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
1-(4-methyl-1,3-thiazole-5-carbonyl)-4-(2-methylphenoxy)piperidine
4-benzyl-3-ethyl-1-(1,2-oxazole-3-carbonyl)-1,4-diazepan-5-one
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
1-methyl-3-{6-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}pyrrolidin-2-one
1-[2-(pyridin-3-yl)piperidin-1-yl]-2-(2,3,6-trimethylphenoxy)ethan-1-one
1-(2-cyclopropylphenyl)-3-[2-(1-hydroxycyclopentyl)ethyl]-3-methylurea
1-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]-3-methylpyrrolidin-2-one
1,5,6-trimethyl-N-[3-(methylamino)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-methyl-N-(3-methylbutyl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
3-(4-methyl-1,3-thiazol-5-yl)-N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]propanamide
3-benzyl-5-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1H-1,2,4-triazole
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
3-[(2-fluorophenyl)formamido]-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide