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4-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-N,N-dimethylaniline
1,3-dimethyl-5-({[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]-2,3-dihydro-1-benzofuran-2-carboxamide
2-{[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-cyclohexyl-N-(2-fluoro-4-methoxyphenyl)-1,4-diazepane-1-carboxamide
8-[(3,4-dimethoxyphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)pyridazine-4-carboxamide
N-{2-[(2-methyl-1-benzofuran-5-yl)formamido]ethyl}acetamide
1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pent-4-en-1-one
3-(3-chlorobenzoyl)-1-(3,4-difluorobenzenesulfonyl)piperidine
5-(2-chlorophenyl)-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]furan-2-carboxamide
N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}propanamide
1-(dimethyl-1,3-oxazole-5-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
ethyl 3-benzyl-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1-one
(1S,5R)-N,N-dimethyl-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-sulfonamide
1-{2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-4-methoxyphenyl}-1H-pyrazole
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
2-cyclopropyl-8-(2-ethoxypyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-hydroxy-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}propanamide
(4aS,8aR)-6-(3-methoxypropanoyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-[2-(3-fluorophenyl)acetyl]-1-(4-methylphenyl)piperazin-2-one
6-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}pyridine-3-carboxamide
1-(1H-imidazol-1-ylmethyl)-N-[3-(4-methoxyphenoxy)propyl]-N-methylcyclopropane-1-carboxamide
4-[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]morpholine
1-[1-(cyclohex-1-en-1-yl)ethyl]-3-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
N-[4-({[(5-methoxy-1H-indol-2-yl)methyl]carbamoyl}methyl)phenyl]butanamide
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}ethan-1-one
5-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
5-{2-[2-(2-chloro-6-fluoro-3-methylphenyl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
10-methoxy-5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
7-chloro-3-[({[1-(morpholin-4-yl)cyclohexyl]methyl}amino)methyl]-1-(prop-2-yn-1-yl)-1,2-dihydroquinolin-2-one
7-(2-phenylquinolin-4-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
3-{2,7-diazaspiro[4.5]decane-7-carbonyl}-4,5,6,7-tetrahydro-1-benzofuran-4-one
4-{2,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl}-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-{5-[2-(1,2-oxazolidin-2-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
3-{[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}phenol
3-(2-methoxyethyl)-1-[3-(1H-pyrazol-5-yl)phenyl]-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
3-(2-amino-1,3-thiazol-4-yl)-N-[(5-methylfuran-2-yl)methyl]propanamide
2-chloro-N-(2-{[(6-hydroxy-1,4-oxazepan-6-yl)methyl]amino}ethyl)benzamide
(1R,5S)-N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-methoxyethyl 3-(2-methylfuran-3-amido)azepane-1-carboxylate
3-[(3R,4S)-1-(1H-imidazol-2-ylmethyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-({3-methyl-7-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
2-(3-methoxyphenyl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-(3-{[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]methyl}phenyl)ethan-1-one
(1S,5R)-6-(cyclopropylmethyl)-3-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S)-2-{[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]amino}propanamide
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-(2-methylphenyl)-1,4-diazepane