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N-[(3-chlorophenyl)methyl]-2-[(isoquinolin-5-yloxy)methyl]-N-methyl-1,3-oxazole-4-carboxamide
1-(3-chloro-4-methoxybenzoyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
2-[(4aR,7aS)-4-[(3-methylpyridin-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridin-2-one
N-[(4-chlorophenyl)methyl]-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
{3-[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]phenyl}methanol
N-ethyl-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
N-[2-(benzylsulfanyl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-(azetidine-1-carbonyl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]benzene-1-sulfonamide
2-(1H-indol-5-yl)-6,7-dimethoxyquinazolin-4-amine
N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
1-methyl-3-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
2-(4-{4-[(4-fluorophenyl)methyl]-2,5-dioxoimidazolidin-4-yl}piperidin-1-yl)pyridine-3-carboxamide
[1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-2,5-dihydro-1H-pyrrol-2-yl]methanol
methyl 4-oxo-4-(3-{[(4-phenylphenyl)formamido]methyl}piperidin-1-yl)butanoate
N-(furan-2-ylmethyl)-2-(2-phenyl-1H-imidazol-1-yl)-N-(pyridin-2-ylmethyl)acetamide
(5S,9aS,9bS)-5-(6-methoxy-2H-chromen-3-yl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-N-(2-methylpropyl)aniline
9-(oxane-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(1S,5R)-3-[2-(3-hydroxyphenyl)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-ethylpyrimidin-2-amine
N-(1,3-benzothiazol-2-yl)-3-[4-(3-cyanopyrazin-2-yl)piperazin-1-yl]propanamide
ethyl 2-{4-[(2-methoxypyridin-3-yl)methyl]piperazin-1-yl}pyridine-3-carboxylate
1-(2-chloropyridin-3-yl)-3-[(3R)-pyrrolidin-3-yl]urea
2-{imidazo[1,2-b]pyridazin-3-yl}-N,N-bis(propan-2-yl)benzamide
2-[(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]hexanamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(3-methoxyphenyl)acetamide
2-[methyl(pyridin-4-ylmethyl)amino]-N-[(4-phenyloxan-4-yl)methyl]acetamide
{1-[6-(dimethylamino)pyrimidin-4-yl]-3-(2-phenoxyethyl)piperidin-3-yl}methanol
2-(methylsulfanyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]benzamide
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]pent-4-enamide
7-(1,3-benzothiazol-2-yl)-4-(3-methoxybenzoyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-(benzyloxy)-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1H-pyrazole-4-carboxamide
N-(3-methylphenyl)-3-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}propanamide
3-({[(1-acetylpiperidin-4-yl)methyl]amino}methyl)-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
2-methoxy-N-{1-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
2-methoxy-5-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)phenol
5-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl})methylamine
(1R,2S,9R)-11-(5-propyl-1,2-oxazole-3-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
6-methyl-2-[2-(1-methylpyrrolidin-3-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxylic acid
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-(2-methoxyethoxy)ethan-1-one
4-{5-[(4-benzylpiperidin-1-yl)methyl]-1,2-oxazole-3-carbonyl}piperazin-2-one
({6-methyl-2-[(2-methylphenyl)methoxy]quinolin-3-yl}methyl)[(3-methyloxetan-3-yl)methyl]amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(pyridin-2-ylmethyl)piperidin-4-amine
4-methyl-1-{[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl}-1,4-diazepan-5-one