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N-(dimethyl-1H-1,2,4-triazol-3-yl)-3-(propoxymethyl)pyrrolidine-1-carboxamide
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(thiophene-2-sulfonyl)piperidine
4-[7-(3-methylfuran-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]thiomorpholine
5,6-dimethyl-3-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-ethyl-4-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-thiazole-5-carboxamide
4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
2-(3,4-dichlorophenyl)-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]morpholine
methyl 4-(4-{2-[(3-methylphenyl)carbamoyl]ethyl}piperidin-1-yl)-4-oxobutanoate
ethyl 4-[(4-methoxyphenyl)methyl]-1-(quinoxaline-5-carbonyl)piperidine-4-carboxylate
N-{[1-(phenoxymethyl)cyclopropyl]methyl}cyclopentanamine
4-(4-methylpiperazin-1-yl)-6-[3-(methylsulfanyl)phenyl]pyrimidin-2-amine
3-phenyl-1-(5-propyl-1,2-oxazole-4-carbonyl)piperazine
3-(ethoxymethyl)-1-methyl-5-[2-(methylsulfanyl)phenyl]-1H-1,2,4-triazole
1-cyclopentyl-4-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperazin-2-one
3-({[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propan-1-ol
[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]bis(1,3-oxazol-4-ylmethyl)amine
2-hydroxy-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
4-(1H-indol-2-ylmethyl)-9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-ethyl-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyrimidine-5-carboxamide
3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-cyclohexanecarbonylpiperidine
N-[(2R,3R)-2-methoxy-1'-(1-methyl-1H-indole-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
4-methyl-6-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
7'-methoxy-1,3',4',5,6,7-hexahydro-1'H-spiro[imidazo[4,5-c]pyridine-4,2'-naphthalene]
N-[(4-methoxypyridin-2-yl)methyl]-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
5-methyl-4-{[1-(1-methyl-1H-pyrazol-5-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
1-(1,1-dioxo-1λ6-thiolan-3-yl)-N-[(5-methylfuran-2-yl)methyl]piperidine-4-carboxamide
1-[4-(difluoromethoxy)-2-methylphenyl]-3-[(3-methyloxetan-3-yl)methyl]urea
1-[(1-{6-[(2-methylbutyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
8-chloro-2-({4-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)quinolin-4-ol
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidine
(3S,4S)-1-[(2,4-diethoxy-3-methylphenyl)methyl]-4-(dimethylamino)pyrrolidin-3-ol
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]-1,4-diazepane
N-(2,5-difluoro-4-hydroxyphenyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
4-(5-methylpyridin-2-yl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-4-ol
N-[4-fluoro-3-(trifluoromethyl)phenyl]-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
14-(5-chloro-2,4-dimethoxyphenyl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(3S,4R)-4-(2-methoxyphenyl)-1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}pyrrolidine-3-carboxylic acid
N-({8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methylpropanamide
N-[2-(ethanesulfonyl)ethyl]-4-(piperidin-3-yl)benzamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
{3-[(4-fluorophenyl)methyl]-1-(9H-purin-6-yl)piperidin-3-yl}methanol
N-[2-(3,4-dimethoxyphenyl)propan-2-yl]-4-methyl-1H-imidazole-5-carboxamide
N-(1,4-oxazepan-6-ylmethyl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
3-fluoro-N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-4-carboxamide
[(2S,6S)-4-(5-methyl-1H-indazole-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
5-methyl-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[(3,4-dimethoxyphenyl)methyl]-2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}acetamide
(3R,4R)-1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
methyl 8-[(2,3-difluorophenyl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate