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1,3-dimethyl-6-(pyridin-3-yl)-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-6-methoxy-N-methylpyrimidin-4-amine
4-{1-[(2-aminopyridin-3-yl)methyl]piperidin-3-yl}benzoic acid
(3S,4R)-1-[(3,4-difluorophenyl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
3-{3-[2-(methylsulfanyl)ethyl]-5-[2-(pyridin-3-yl)ethyl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-2-(hydroxymethyl)piperidine-1-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
3-chloro-N-cyclopentyl-4-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide
{3-[(E)-2-phenylethenyl]phenyl}methanamine
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-methyl-1,3-thiazole-4-carboxamide
3-(4-hydroxyphenyl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
6-ethyl-2-methyl-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]quinoline
1-cyclopentyl-4-({[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](methyl)amino}methyl)pyrrolidin-2-one
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[(dimethylamino)methyl]piperidin-4-ol
3-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-2-(1H-imidazol-2-yl)benzamide
1-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-4-{5-[(4-methylphenyl)sulfanyl]furan-2-yl}-1H-1,2,3-triazole
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-[2-({[4-(1H-pyrazol-4-yl)phenyl]carbamoyl}amino)ethyl]piperidine-3-carboxamide
methyl 5-{3-cyclobutyl-6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-2-hydroxybenzoate
3-[(propan-2-yl)sulfamoyl]-5-(1H-1,2,4-triazol-1-yl)benzoic acid
N-cyclopropyl-2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
1-[4-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)-1,4-diazepan-1-yl]ethan-1-one
(1R,3S)-3-methoxy-7-[6-(methoxymethyl)pyridine-2-carbonyl]-7-azaspiro[3.5]nonan-1-ol
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-(1-cyclopropylethyl)pyridin-2-amine
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}({[2-(trifluoromethoxy)phenyl]methyl})amine
N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
3-(5-{1-[(2,6-difluoro-3-methylphenyl)methyl]-1H-imidazol-2-yl}thiophen-2-yl)prop-2-yn-1-ol
2-{3-[2-methyl-6-(trifluoromethyl)pyridin-3-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrazine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(methylamino)-1,3-thiazole-4-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(2-methoxypyrimidin-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
N-cyclopropyl-1-(1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)piperidine-3-carboxamide
1-[2-(3-chlorophenyl)ethyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
1-(2-oxo-2-{4-[2-(pyridin-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethyl)-4-phenylpyrrolidin-2-one
2,4-dimethyl-6-{3-[3-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}pyrimidine
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
N-{1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]methyl}-3,5-dimethoxybenzoic acid
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-[4-(ethylsulfanyl)phenyl]-3-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}urea
3-(2-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)pyrrolidine
N-tert-butyl-2-(1-methyl-6-oxo-1,6-dihydropyridazin-3-yl)benzene-1-sulfonamide
1-(5-methylthiophene-2-carbonyl)-N-(2-phenylethyl)piperidine-4-carboxamide
2-amino-6-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
2,3-dimethyl-N-({1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}methyl)benzamide
6-ethyl-N-[2-hydroxy-1-(thian-4-yl)ethyl]-2-methylquinoline-4-carboxamide
{3-[(3-chlorophenyl)methyl]-1-(pyrimidin-2-yl)piperidin-3-yl}methanol